• NEBANNER

4-chloro-n- (4,5-dihydro-1h-imidazol-2-yl) -6-methoxy-2-methyl-5-pyrimidinamin;

4-chloro-n- (4,5-dihydro-1h-imidazol-2-yl) -6-methoxy-2-methyl-5-pyrimidinamin;

Takaitaccen Bayani:

Tsarin kwayoyin halitta: C9H12ClN5O

Nauyin Kwayoyin: 241.677

Saukewa: 75438-57-2


Cikakken Bayani

Tags samfurin

Aikace-aikace

Yana aiki ta hanyar ƙarfafa tsakiyar presynaptic alpha 2- masu karɓa.Tasirinsa yana kama da nifedipine, mai adawa da calcium, da captopril, mai hana ACE.Don mahimmancin hauhawar jini.

Ya kamata wannan samfurin ya ɗauki ƙa'idar magani na mutum ɗaya.Gabaɗaya farawa daga mafi ƙarancin kashi, wato, 0.2mg, sau ɗaya a rana, ana sha da safe.Ya kamata a yi gyare-gyaren sashi a cikin tazara na makonni uku har sai an sami sakamako mai gamsarwa.Maganin da aka saba shine 0.2mg sau ɗaya, sau biyu a rana (safe da maraice).Matsakaicin adadin kowane lokaci ba zai wuce 0.4mg ba, kuma matsakaicin adadin yau da kullun ba zai wuce 0.6mg ba.Ga marasa lafiya tare da ƙarancin ƙarancin koda ko matsakaici, kashi ɗaya bai kamata ya wuce 0.2 MG ba ko adadin yau da kullun kada ya wuce 0.4 MG.

Wannan samfurin agonist na α2-receptor, wanda shine maganin antihypertensive imidazoline.Ana amfani da shi don matsakaici da matsananciyar hauhawar jini na farko da na sakandare.

Domin yana hana fita da motsi na gastrointestinal tract, kuma ya dace da masu fama da hauhawar jini masu fama da cutar ulcer.Haɗin wannan magani da diuretics na iya inganta haɓakar inganci sosai.Magani ne na tsakiya mai ƙarfi na maganin hauhawar jini da kuma magani na antihypertensive na layi na biyu.An fi gudanar da shi a cikin gida a cikin ilimin ophthalmology.Wannan samfurin yana da tasirin rage matsa lamba na intraocular, kuma baya shafar almajiri da tsarin daidaita idanu.Yana iya takure magudanar jini a cikin ido, rage samar da jin dadi, da cimma tasirin rage matsa lamba na intraocular.Yana fara yin tasiri bayan mintuna 15 bayan saukar ido kuma yana iya kula da tasirin kusan awanni 8.

Standard:EP10
Abubuwan bincike:97.5-102.0%

Na waje:Fari ko kusan yayin foda
Kunshin:1kg/bag ko kamar yadda abokan ciniki suka bukata

Layin Samfuri mai haɗaka da albarkatu

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Takaddun shaida

JIN DUN Medical yaCancantar ISO kuma ya cika ka'idodin samar da GMP, ƙwararrun ƙwararrun haɗaɗɗun ƙwayoyi na cikin gida da na waje tare da ƙwararrun ƙwarewa don jagorantar R&D na kamfani.

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Abũbuwan amfãni a kan Gyaran Likita

TECHNOL OGY AMFANIN
●High Matsi Catalytic Hydrogenation.Babban Matsi na Hydrogenolysis Reaction.Maganin Cryogenic (<-78% C)
●Aromatic Heterocyclic Synthesis
●Maganar Sake Shiryawa
●Matsalar Chiral
●Heck, Suzuki,Negishi,Sonogashira .Gignard Reaction

JIN DUN R&D

Kayan aiki

Our Lab yana da daban-daban na gwaji da kuma gwaji kayan aiki, kamar: NMR (Bruker 400M), HPC, Chiral-HPLC, LC-MS, LC-MS/MS (API 4000) , IR, UV, GC, GC-MS, Chromatography, Microwave Synthesizer, Parallel Synthesizer, Bambance-bambancen Scanning Calorimeter (DSC), Electron Microscope...

Ƙungiyar R&D

Jindun Medical yana da rukuni na ƙwararrun ma'aikatan R&D, kuma yana ɗaukar ƙwararrun masana harhada magunguna na cikin gida da na waje don jagorantar R&D, yana sa ƙirarmu ta fi dacewa da inganci.

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Raba Harka

Mun taimaka wa manyan kamfanonin harhada magunguna na cikin gida da yawa, kamarHansoh, Hengrui da HEC Pharm.Anan zamu nuna sashinsu.

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Hali na Farko na Farko:

Lambar Waya: 110351-94-5

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Hali na Musamman na Biyu:

Lambar Waya: 144848-24-8

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Halin Hali na Uku:

Lambar Waya: 200636-54-0

Yanayin Haɗin kai

1.Keɓance Sabbin Matsakaici ko APIs.Daidai da raba shari'ar na sama, abokan ciniki suna da buƙatun takamaiman Matsakaici ko APIs, kuma ba za su iya samun samfuran da ake buƙata ba a kasuwa, sannan za mu iya taimakawa don Keɓancewa.

2.Haɓaka Tsari don Tsofaffin Kayayyaki.Ƙungiyarmu za ta taimaka don ingantawa da haɓaka irin wannan samarwa wanda hanyar amsawa ta tsufa, farashin samarwa yana da yawa, kuma ingancin ya yi ƙasa.Za mu iya samar da cikakkun takardun shaida don canja wurin fasaha da haɓaka tsari, taimakawa abokin ciniki don samar da ingantaccen aiki.

Daga maƙasudin miyagun ƙwayoyi zuwa INDs, JIN DUN Medical yana ba kumafita na R&D keɓaɓɓen tsayawa ɗaya tasha.

JIN DUN Medical ya dage kan ƙirƙirar ƙungiyar tare da mafarkai, yin samfura masu daraja, ƙwararrun ƙwararrun ƙwararrun ƙwararrun ƙwararrun ƙwararrun ƙwararrun ƙwararrun ƙwararrun ƙwararrun ƙwararrun ƙwararrun ƙwararrun ƙwararrun ƙwararrun ƙwararrun ƙwararrun ƙwararrun ƙwararrun ƙwararrun ƙwararrun ƙwararrun ƙwararrun ƙwararrun ƙwararrun ƙwararrun ƙwararrun ƙwararrun ƙwararrun ƙwararrun ƙwararrun ƙwararrun ƙwararrun ƙwararrun ƙwararrun ƙwararrun ƙwararrun ƙwararrun ƙwararrun ƙwararrun ƙwararrun ƙwararrun ƙwararrun ƙwararrun ƙwararrun ƙwararrun ƙwararrun ƙwararrun ƙwararrun ƙwararrun ƙwararrun ƙwararrun ƙwararrun ƙwararrun ƙwaƙƙwaran, masu tsattsauran ra'ayoyi, masu tsauri, da kuma fita gabaɗaya don zama amintaccen abokin tarayya kuma abokin abokan ciniki!


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