5,6,7,7a-tetrahydrothieno(3,2-c) pyridine-2(4h) hydrochloride daya

5,6,7,7a-tetrahydrothieno(3,2-c)pyridine-2(4h) -ana amfani da hydrochloride daya a matsayin tsaka-tsakin Prasugrel.

Prasugrel wani thiophenopyridine antiplatelet ne wanda Eli Lilly da daiichisankyo, wani masana'antar harhada magunguna ta Japan suka kirkira.Magani ne na farko.Yana samar da kwayar halitta mai aiki bayan metabolism ta hanyar cytochrome P450 a cikin hanta kuma yana haɗuwa tare da mai karɓar platelet P2Y12 don yin aiki mai ƙarfi a kan haɗuwar platelet.Nazarin asibiti sun tabbatar da cewa kashi 60 na MG yana da mafi kyawun tasirin anticoagulant fiye da 300 MG daidaitaccen kashi da 600 MG ya karu kashi na clopidogrel, wanda zai iya rage haɗarin bugun zuciya, bugun jini da mutuwa saboda cututtukan zuciya da kashi 20%, kuma yana da saurin tasiri. , Kyakkyawan maganin warkewa, kyakkyawan juriya na miyagun ƙwayoyi da bioavailability, da ƙarancin guba.